
Brimonidine Tartrate
CAS No. 70359-46-5
Brimonidine Tartrate( AGN 190342LF | Alphagan P )
Catalog No. M15704 CAS No. 70359-46-5
Brimonidine Tartrate is a highly selective α-adrenergic receptor agonist with EC50 of 0.45 nM for the α2A adrenoreceptor, and used to treat open-angle glaucoma or ocular hypertension.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
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500MG | 113 | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameBrimonidine Tartrate
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NoteResearch use only, not for human use.
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Brief DescriptionBrimonidine Tartrate is a highly selective α-adrenergic receptor agonist with EC50 of 0.45 nM for the α2A adrenoreceptor, and used to treat open-angle glaucoma or ocular hypertension.
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DescriptionBrimonidine Tartrate is a highly selective α-adrenergic receptor agonist with EC50 of 0.45 nM for the α2A adrenoreceptor, and used to treat open-angle glaucoma or ocular hypertension.(In Vitro):[3H]Brimonidine (UK 14304) is a full agonist at alpha 2-adrenergic receptors. [3H]Brimonidine (UK 14304) labels at least 2 specific binding sites in human brain that both have the characteristics of an alpha 2-adrenergic binding site. GTP decreases agonist binding at both of these sites, but with different potencies at each site.
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In Vitro[3H]Brimonidine (UK 14304) is a full agonist at alpha 2-adrenergic receptors. [3H]Brimonidine (UK 14304) labels at least 2 specific binding sites in human brain that both have the characteristics of an alpha 2-adrenergic binding site. GTP decreases agonist binding at both of these sites, but with different potencies at each site [1-3].
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In Vivo——
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SynonymsAGN 190342LF | Alphagan P
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PathwayEndocrinology/Hormones
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TargetAdrenergic Receptor
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Recptorα2A-adrenergic receptor
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Research AreaOther Indications
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Indication——
Chemical Information
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CAS Number70359-46-5
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Formula Weight442.22
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Molecular FormulaC15H16BrN5O6
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Purity>98% (HPLC)
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SolubilityWater: 75 mg/mL (169.59 mM); DMSO: 88 mg/mL (198.99 mM)
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SMILESC1CN=C(N1)NC2=C(C3=NC=CN=C3C=C2)Br.[C@@H]([C@H](C(=O)O)O)(C(=O)O)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.WoldeMussie E, et al. Invest Ophthalmol Vis Sci, 2001, 42(12), 2849-2855.
molnova catalog



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